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García-Cuesta, E. M.; Martínez, P.; Selvaraju, K.; Gómez-Pozo, A.M.; D’Agostino, G.; Gardeta, S.; Quijada-Freire, A.; Blanco-Gabella, P.; Roca, C.; Jiménez-Saiz, R.; García-Rubia, A.; Soler-Palacios, B.; Lucas, P.; Ayala-Bueno, R.; Santander-Acerete, N.; Carrasco, Y.R.; Martínez, A.; Campillo, N. E.; Jenssen, L.; Rodríguez-Frade, J. M.; Santiago, C.; Mellado, M.
[2024]. Allosteric modulation of the CXCR4:CXCL12 axis by targeting receptor nanoclustering via the TMV-TMVI domain. eLife, 2024, https://doi.org/10.7554/eLife.93968.1
Cuevas, E. P.; Martinez-Gonzalez, L.; Gordillo, C.; Tosat-Bitrián, C.; Pérez de la Lastra, C.; Sáenz, A.; Gil, C.; Palomo, V.; Martin-Requero, A.; Martinez, A.
[2024]. Casein kinase 1 inhibitor avoids TDP-43 pathology propagation in a patient-derived cellular model of amyotrophic lateral sclerosis. Neurobiol Dis 2024, 192, 106430
Etxebeste-Mitxeltorena, M.; Niza, E.; Martinez-Fajardo, C.; Gil, C.; Gómez-Gómez, L.; Martinez, A.; Ahrazem, O.
[2024]. Neuroprotective properties of exosomes and chitosan nanoparticles of Tomafran, a bioengineered tomato enriched in crocins. Nat Prod Bioprospect 2024, 14, 9
Benítez-Fernández, R.; Josa-Prado, F.; Sánchez, E.; Lao, Y.; García-Rubia, A.; Cumella, J.; Martínez, A.; Palomo, V.; de Castro, F.
[2024]. Efficacy of a benzothiazole-based LRRK2 inhibitor in oligodendrocyte precursor cells and in a murine model of multiple sclerosis. CNS Neurosci Ther 2024, 30, e14552
Atienza-Navarro, I.; del Marco, A.; Alves-Martinez, P.; Garcia-Perez, A.; Raya-Marin, A.; Benavente-Fernandez, I.; Gil, C.; Martinez, A.; Lubian-Lopez, S.; Garcia-Alloza, M.
[2024]. Glycogen synthase kinase-3β inhibitor VP3.15 ameliorates neurogenesis, neuronal loss and cognitive impairment in a model of germinal matrix- intraventricular hemorrhage of the preterm newborn. Transl Stroke Res 2024, doi 10.1007/s12975-023-01229-2
Garcia-Rubia, A.; Lasala, F.; Ginex, T.; Morales-Tenorio, M.; Olal, C.; Heung, M.; Oquist, P.; Galindo, I.; Cuesta-Geijo, M.; Casasnovas, J. M.; Campillo, N. E.; Canales, Á.; Alonso, C.; Martínez, A.; Muñoz-Fontela, C.; Delgado, R.; Gil, C.
[2023]. N'-Phenylacetohydrazide derivatives as potent Ebola virus entry inhibitors with an improved pharmacokinetic profile. J Med Chem 2023, 66, 8, 5465-5483
Martinez-Gonzalez, L.; Cuevas, E. P.; Tosat, C.; Nozal, V.; Gil, C.; Palomo, V.; Martin-Requero, A.; Martinez, A.
[2023]. TTBK1 and CK1 inhibitors restore TDP-43 pathology and avoid disease propagation in lymphoblast from Alzheimer's disease patients. Front Mol Neurosci 2023, 16, 1243277
Rabanal Basalo, A.; Navarro Pablos, M.; Viejo Pinero, N.; Vila Méndez, M. L.; Molina Barcena, V.; Montilla Bernabé, A.; Villanueva Morán, M. D. P.; Blanco Gallego, A. M.; Guirao Sánchez, C.; Juárez Antón, S.; Fernández Rodríguez, Á.; Revuelta Puigdollers, M. L.; Sarriá Sánchez, M. T.; Martín Alegre, C.; Martínez Álvarez, M.; Mestre de Juan, M.; Mielgo Salvador, R.; Gijón Seco, M. T.; Saníger Herrera, J. M.; Rodríguez Jiménez, M. E.; Navas de la Peña, B.; Santa Cruz Hernández, J.; Abad Esteban, A. M.; Díaz Martín, R.; García Pérez, L.; Herrero Vanrell, P.; Arias de Saavedra Criado, M. I.; Vaquero Vinent, A.; López Gómez, V.; Montegrifo Rentero, V. M.; Simón Miguel, L.; Campo Martos, I.; Ortiz Zamorano, S.; Izquierdo Zamarriego, M. J.; Vázquez Carrión, I.; López Valero, R. M.; Gil, C.; Martínez, A.; Soler López, B.
[2023]. A randomized, double-blind study on the efficacy of oral domperidone versus placebo for reducing SARS-CoV-2 viral load in mild-to-moderate COVID-19 patients in primary health care. Ann Med 2023, 55, 2268535
Jing, L.; Wei, W.; Meng, B.; Chantegreil, F.; Nachon, F.; Martínez, A.; Wu, G.; Zhao, H.; Song, Y.; Kang, D.; Brazzolotto, X.; Zhan, P.; Liu, X.
[2023]. Rapid discovery and crystallography study of highly potent and selective butylcholinesterase inhibitors based on oxime-containing libraries and conformational restriction strategies. Bioorg Chem 2023, 134, 106465
Rodríguez-Periñán, G.; de la Encarnación, A.; Moreno, F.; López de Munain, A.; Martínez, A.; Martín-Requero, Á.; Alquézar, C.; Bartolomé, F.
[2023]. Progranulin deficiency induces mitochondrial dysfunction in frontotemporal lobar degeneration with TDP-43 inclusions. Antioxidants, 2023, 12, 581
Zheng, Y.; Schroeder, S.; Kanev, G. K.; Botros, S. S.; William, S.; Sabra, A.-N. A.; Maes, L.; Caljon, G.; Gil, C.; Martinez, A.; Salado, I. G.; Augustyns, K.; Edink, E.; Sijm, M.; de Heuvel, E.; de Esch, I. J. P.; van der Meer, T.; Siderius, M.; Sterk, G. J.; Brown, D.; Leurs, R.
[2023]. To target or not to target Schistosoma mansoni cyclic nucleotide phosphodiesterase 4A? Int J Mol Sci 2023, 24, 6817
Vila Méndez, M. L.; Antón Sanz, C.; Cárdenas García, A. D. R.; Bravo Malo, A.; Torres Martínez, F. J.; Martín Moros, J. M.; Real Torrijos, M.; Vendrell Covisa, J. F. J.; Guzmán Sierra, O.; Molina Barcena, V.; Viejo Pinero, N.; Fernández Díaz, C.; Arroyo Burguillo, P.; Blanco Gallego, A. M.; Guirao Sánchez, C.; Montilla Bernabé, A.; Villanueva Morán, M. D. P.; Juárez Antón, S.; Fernández Rodríguez, Á.; Somoza Calvo, M.; Cerrada, E. C.; Pérez Mañas, G.; Sánchez Calso, A.; Vallejo Somohano, F.; Cauqui Díaz, C.; Viñas Fernández, G.; Molina París, J.; González Godoy, M.; Lumbreras García, G.; Rosado Martín, J.; Rodríguez Hernández, A.; López Antúñez, S.; Vázquez Perfecto, G.; Marcello Andrés, M. C.; Puente García, N. M.; Gil, C.; Martínez, A.; Soler López, B.
[2023]. Efficacy of bromhexine versus standard of care in reducing viral load in patients with mild-to-moderate COVID-19 disease attended in primary care: A randomized open-label trial. J Clin Med 2023, 12, 142.
Staderini, M.; Vanni, S.; Baldeschi, A. C.; Giachin, G.; Zattoni, M.; Celauro, L.; Ferracin, C.; Bistaffa, E.; Moda, F.; Pérez, D. I.; Martínez, A.; Martín, M. A.; Martín-Cámara, O.; Cores, Á.; Bianchini, G.; Kammerer, R.; Menéndez, J. C.; Legname, G.; Bolognesi, M. L.
[2023]. Bifunctional carbazole derivatives for simultaneous therapy and fluorescence imaging in prion disease murine cell models. Eur J Med Chem 2023, 245, 114923
Liu, Z.; Li, A.; Ali, T.; He, K.; Gao, R.; Liufang, H.; Qiang, H.; Li, T.; Li, N.; Garcia, A.; Gil, C.; Martinez, A.; Lipina, T. V.; Li, S.
[2023]. Neuronal lack of PDE7a disrupted working memory, spatial learning, and memory but facilitated cued fear memory in mice. Prog Neuropsychopharmacol Biol Psychiatry 2023, 120, 110655